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Fragment-based drug discovery

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Acknowledgments

I am grateful to Rod Hubbard of Vernalis and Mark Murko of Vertex for giving balanced answers to my many challenging questions and to David Bailey of IOTA Pharmaceuticals [22] for helping me with Table 1. I would also like to thank several people who have given me ideas but wished to remain anonymous.

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Correspondence to Wendy A. Warr.

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Warr, W.A. Fragment-based drug discovery. J Comput Aided Mol Des 23, 453–458 (2009). https://doi.org/10.1007/s10822-009-9292-1

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